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2000
Volume 3, Issue 4
  • ISSN: 1568-0266
  • E-ISSN: 1873-4294

Abstract

In this review the latest developments in ligand design for the adenosine A1 receptor are summarized. Novel series of agonists and antagonists are discussed, leading to the conclusion that ligands truly selective for the human adenosine A1 receptor are still scarce.

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/content/journals/ctmc/10.2174/1568026033392165
2003-02-01
2025-06-19
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  • Article Type:
    Review Article
Keyword(s): adenosine receptor; affinity; intrinsic activity; medicinal chemistry
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